|
[1]
|
Kormis, G. (1984) 1,3,4-thiadiazoles. In: A. R. Katritzky, Ed., Comprehensive Heterocyclic Chemistry, Pergamon Press, 6, 545-578.
|
|
[2]
|
Hussein, M.A., Kafafy, A.H.N., Abdel-Moty, S.G. and Abou-Ghadir, O.M.F. (2009) Synthesis and biological activities of new substituted thiazoline-quinoline derivatives. Acta Pharmaceutica, 59, 365-382.
doi:10.2478/v10007-009-0033-8
|
|
[3]
|
Pintilie, O., Profire, L., Sunel, V., Popa, M. and Pui, A. (2007) Synthesis and antimicrobial activity of some new 1,3,4-thiadiazole and 1,2,4-triazole compounds having a D,L-methionine moiety. Molecules, 12, 103-113.
doi:10.3390/12010103
|
|
[4]
|
Faroumadi, A., Mirzaei, M. and Shafiee, A. (2001) Antitubercular agents, I: Synthesis and antituberculosis activity of 2-aryl-1,3,4-thiadiazole derivatives. Pharmazie, 56, 610-612.
|
|
[5]
|
Mamolo, M.G., Falagiani, V., Zanpier, D., Vio, L. and Banfi, F. (2001) Synthesis and antimycobacterial activity of [5- (pyridin-2-yl)-1,3,4-thiadiazol-2-ylthio]acetic acid arylidene- hydrazide derivatives. II Farmaco, 56, 587- 592. doi:10.1016/S0014-827X(01)01097-7
|
|
[6]
|
Zou, X.J., Lai, L.H., Jin, G.Y. and Zhang, Z.X. (2002) Synthesis, fungicidal activity, and 3D-QSAR of pyridazinone-substituted 1,3,4-oxadiazoles and 1,3,4-thiadiazoles. Journal of Agricultural and Food Chemistry, 50, 3757-3760. doi:10.1021/jf0201677
|
|
[7]
|
Chen, H., Li, Z. and Han, Y. (2000) Synthesis and fungicidal activity against rhizoctonia solani of 2-alkyl (alkylthio)-5-pyrazolyl-1,3,4-oxadiazoles (thiadiazoles). Journal of Agricultural and Food Chemistry, 48, 5312-5315.
doi:10.1021/jf991065s
|
|
[8]
|
Clerici, F., Pocar, D., Guido, M., Loche, A., Perlini, V. and Brufani, M. (2001) Synthesis of 2-amino-5-sulfanyl- 1,3,4-thiadiazole derivatives and evaluation of their antidepressant and anxiolytic activity. Journal of Medicinal Chemistry, 44, pp. 931-936.
doi:10.1021/jm001027w
|
|
[9]
|
Palaska, E., Sahin, G., Kelincen, P., Durlu, N.T. and Altionax, G. (2002 ) Synthesis and anti-inflammatory activity of 1-acylthiosemicarbazides, 1,3,4-oxadiazoles, 1,3, 4-thiadiazoles and 1,2,4-triazole-3-thiones. II Farmaco, 57, 101-107. doi:10.1016/S0014-827X(01)01176-4
|
|
[10]
|
Shenone, S., Bruno, O., Ranise, A., Bondavalli, W., Falcone, G., Giordano, L. and Vitelli, M. (2001) 3-Arylsulphonyl-5-arylamino-1,3,4-thiadiazol-2(3H) ones as anti- inflammatory and analgesic agents. Bioorganic & Medicinal Chemistry, 9, 2149-2153.
doi:10.1016/S0968-0896(01)00121-3
|
|
[11]
|
Onko., T. Cakir, B. and Sahin, M.F. (2004) Synthesis and antinociceptive activity of 2-[(2-Oxobenzothiazolin-3-yl) methyl]-5-aminoalkyl/aryl-1,3,4-thiadiazole. Turkish Journal of Chemistry, 28, 461-468.
|
|
[12]
|
Azab, M.E., El-Hag Ali, G.A.M. and Abd El-Wahab, A.H.F. (2003) Studies on thiazolopyridines: A novel synthesis of bisthiazolopyridines as promising antimicrobial agents. Acta Pharmaceutica, 53, 213-221.
|
|
[13]
|
Sondhi, S.M., Singh, N., Lahoti, A.M., Bajaj, K., Kumar, A., Lozach, O. and Meijer, L. (2005) Synthesis of acridinyl-thiazolino derivatives and their evaluation for anti-inflammatory, analgesic and kinase inhibition activities. Bioorganic & Medicinal Chemistry, 13, 4291-4299.
doi:10.1016/j.bmc.2005.04.017
|
|
[14]
|
Mahler, G., Serra, G., Dematteis, S., Saldana, J., Dominguez, L. and Manta, E. (2006) Synthesis and biological evaluation of simplified mycothiazole analogues. Bioorganic & Medicinal Chemistry Letters, 16, 1309- 1311. doi:10.1016/j.bmcl.2005.11.072
|
|
[15]
|
Shih, M. and Ke, F. (2004) Syntheses and evaluation of antioxidant activity of sydnonyl substituted thiazolidinone and thiazoline derivatives. Bioorganic & Medicinal Chemistry Letters, 12, 4633-4643.
doi:10.1016/j.bmc.2004.06.033
|
|
[16]
|
Godefroi, E.F. and Platje, J.Th. (1972) DL-1- (.alpha.-Methylbenzyl)-2-methylimidazole-5-carboxylate esters. Synthesis and pharmacological properties. Journal of Medicinal Chemistry, 15, 336-337.
doi:10.1021/jm00273a035
|
|
[17]
|
Harfenist, M., Soroko, F.E. and Mckenzie, G.M. (1978) 2-(Alkoxyaryl)-2-imidazoline monoamine oxidase inhibitors with antidepressant activity. Journal of Medicinal Chemistry, 21, 405-409.
doi:10.1021/jm00202a021
|
|
[18]
|
Kornicka, A., Hudson, A.L. and Bednarski, P.J. (2009) Synthesis and biological activity of some 2-imidazolinylhydrazone derivatives. Acta Poloniae Pharmaceutica-Drug Research, 66, 523-534.
|
|
[19]
|
Desai, N.C., Bhavsar, A.M. and Baldaniya, B.B. (2009) Synthesis and antimicrobial activity of 5-imidazolinone derivatives. Journal of Postgraduate Medicine, 71, 90- 94.
|
|
[20]
|
Solankee, A., Kapadia, K., Thakor, I., Patel, J. and Lad, S. (2004) Synthesis and Antimicrobial Activity of 1-(4′ -Trifluoro methylphenyl and- 2-phenyl-4-(benzylidene/ substituted Benzylidene/2’ furylidene/2’-thienylidene)- imidazolin-5-ones. Asian Journal of Chemistry, 16, 917- 920.
|
|
[21]
|
Mor, M., Bordi, F., Silva, C., Rivara, S., Zuliani, V., Vacodio, F., Morini, G., Barocelli, E., Ballabeni, V., Impicciatore, M. and Plazzi, P.V. (2000) Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups. II Farmaco, 55, 27-34.
doi:10.1016/S0014-827X(99)00115-9
|
|
[22]
|
Giorgioni, G., Claudi, F., Ruggieri, S., Ricciutelli, M., Palmieri, G.F., Di-Stefano, A., Sozio, P., Cerasa, L.S., Chiavaroli, A., Ferrante, C., Orlando and G., Glennon, (2010) Design, synthesis, and preliminary pharmacological evaluation of new imidazolinones as l-DOPA prodrugs. Bioorganic & Medicinal Chemistry Letters, 18, 1834-1843. doi:10.1016/j.bmc.2010.01.041
|
|
[23]
|
Abunada, N.M., Hassaneen, H.M., Kandile, N.G. and Miqdad, O.A. (2008) Synthesis and biological activity of some new pyrazoline and pyrrolo[3,4-c]pyrazole-4,6- dione derivatives: reaction of nitrilimines with some dipolarophiles. Molecules, 13, 1011-1024.
doi:10.3390/molecules13041011
|
|
[24]
|
Abunada, N.M., Hassaneen, H.M., Kandile, N.G. and Miqdad, O.A. (2008) Synthesis and antimicrobial activity of some new pyrazole, fused pyrazolo[3,4-d]-pyrimidine and pyrazolo[4,3-e][1,2,4]-triazolo[1,5-c]pyrimidine derivatives. Molecules, 13, 1501-1517.
doi:10.3390/molecules13071501
|
|
[25]
|
Abunada, N.M., Hassaneen, H.M., Abu Samaha, A.M. and Miqdad, O.A. (2009) Synthesis and antimicrobial evaluation of some new pyrazole, pyrazoline and chromeno [3,4-c]pyrazole derivatives. Journal of Brazilian Chemical Society, 20, 975-987.
doi:10.1590/S0103-50532009000500024
|
|
[26]
|
Hassaneen, H.M., Shawali, A.S., Khalil, M.S. and Abdallah, T.A.A. (1993) One step synthesis of benzimidazo[2,1-c] [1,2,4]triazole derivatives using hydrazonoyl halides. Heterocycles, 36, 1775-1781.
doi:10.3987/COM-93-6344
|
|
[27]
|
Hassaneen, H.M., Abbas, I.M., Abdelhadi, H.A., Abdallah, T.A. and Algharib, M.S. (1994) Reactions of 5-oxo- 2-pyrazolin-4-thiocarboxanilides and 5-oxo-2-oxazolin- 4-thiocarboxanilides with hydrazonoyl halides. Sulfur Letters, 17, 295-307.
|
|
[28]
|
Hassaneen, H.M., Elwan, N.M., Abdelhadi, H.A. and Abdallah, T.A. (1995) Reactions of thioanilides with active chloromethylene compounds. Synthesis of 1,3- oxathiol-2-ylidene derivatives. Sulfur Letters, 18, 121- 128.
|
|
[29]
|
Hassaneen, H.M., Harhash, A.H.E., Abunada, N.M., Abdallah, T.A. and Algharib, M.S. (1993) Cyano-(1-methylbenzimidazol-2-yl)thioacetanilide in the synthesis of 2,3-dihydro-1,3,4-thiadiazole derivatives. The Journal of Chemical Research, 1993, 194-195.
|
|
[30]
|
Argyropoulou, E.C. and Thessalonikeos, E. (1990) Reactions of nitrile oxides and nitrile imines with 4-arylidene- 2-phenyl-5(4H)-thiazolones. Liebigs Ann. Chemistry, 1097-1100. doi:10.1002/jlac.1990199001198
|
|
[31]
|
Johnson, T.B. and Hadley, S.E. (1915) Researches on hydantoins. XXIX. Geometrical isomerism in the hydantoin series. Journal of American Chemical Society, 37, 171-177. doi:10.1021/ja02270a017
|
|
[32]
|
Wolkoff, P. (1975) A new method of preparing hydrazonyl halides. Canadian Journal of Chemistry, 53, 1333- 1335. doi:10.1139/v75-183
|
|
[33]
|
Hassaneen, H.M., Elwan, N.M., Harhash, A. and Shawali, A.S. (1984) The regioselectivity in the formation of pyrazolines and pyrazoles from nitrile imines. Journal of Heterocyclic Chemistry, 21, 1013-1016.
doi:10.1002/jhet.5570210417
|
|
[34]
|
Hassaneen, H.M., Mousa, H.A.H., Abed, N.M. and Shawali, A.S. (1988) Chemistry of C-Heteroarylhydrazidoyl halides. Synthesis and reactions of n-(p-nitrophenyl)-c- (2-thienyl)-formohydrazidoyl halides. Heterocycles, 27, 695-706. doi:10.3987/COM-87-4381
|
|
[35]
|
Shawali, A.S., Hassaneen, H.M. and Ibrahim, H.A. (1990) Synthesis and cycloaddition reactions of N-aryl-2-furohydrazonoyl chlorides. Archives of Pharmacal Research, 13, 126-131.
doi:10.1007/BF02857788
|
|
[36]
|
Aylward, J.B. and Scott, F.L. (1969) Preparation and sovolysis of N1-arylbenzohydrazonyl bromides. Journal of Chemical Society (B), 1969, 1080-1084.
doi:10.1039/j29690001080
|
|
[37]
|
Eweiss, N.F. and Osman, A. (1980) Synthesis of heterocycles. Part II. New routes to acetylthiadiazolines and alkylazothiazoles. Journal of Heterocyclic Chemistry, 17, 1713-1717. doi:10.1002/jhet.5570170814
|
|
[38]
|
Shawali, A.S., Eweiss, N.F., Hassaneen, H.M. and Algharib, M.S. (1975) Synthesis and rearrangement of ethyl aryloxyglyoxalate arylhydrazones. Bulletin of the Chemical Society of Japan, 48, 365-366.
doi:10.1246/bcsj.48.365
|
|
[39]
|
Shawali, A.S. and Osman, A. (1971) Synthesis and reactions of phenylcarbamoylarylhydrazidic chlorides. Tetrahedron, 27, 2517-2528.
doi:10.1016/S0040-4020(01)90753-7
|
|
[40]
|
Shawali, A.S. and Abdelhamid, A.O. (1976) Reaction of dimethylphenacylsulfonium bromide with N-nitrosoacetarylamides and reactions of the products with nucleophiles. Bulletin of the Chemical Society of Japan, 49, 321-324. doi:10.1246/bcsj.49.321
|
|
[41]
|
Farag, A.M. and Algharib, M.S. (1988) Synthesis and reactions of C-(2-thenoyl)-N-arylformahydrazidoyl bromides. Org. Prep. Procd. Int., 20, 521-526.
doi:10.1080/00304948809356298
|
|
[42]
|
Hassaneen, H.M., Shawali, A.S., Elwan, N.M. and Abunada, N.M. (1992) Reaction of 1-(2-naphthoyl) methyl-2-dimethylsulfonium bromide with N-nitroso-N- arylacetamides and reactions of the products with some nucleophiles. Sulfur Letters, 13, 273-285.
|
|
[43]
|
Huisgen, R., Grashey, R., Seidel, M., Knupfer, H. and Schmidt, R. (1962) 1,3-Dipolare Additionen, III. Umsetzungen des Diphenylnitrilimins mit Carbonyl und Thiocarbonyl-Verbindungen. Just Liebigs Ann. Chemistry, 658, 169-180. doi:10.1002/jlac.19626580115
|
|
[44]
|
Abdelhamid, A.O. and Abdou, S.E. (1987) Reactions of cyanothioacetamide with hydrazidoyl halides: a novel synthesis of some hydrazidoyl sulfides and triazole derivatives. Sulfur Letters, 6, 41-47.
|
|
[45]
|
Mohareb, R.M., Sherif, S.M., Abdel-Aal, F.A.M. and Sayed, N.I.A. (1990) One-pot synthesis of polyfunctionally substituted 2,3-dihydrothiazoles and thiazolidinones. Just Liebigs Ann. Chemistry, 1143-1146.
|