Dr. Joaquín M. Campos
Departamento de Química Farmacéuticay Orgánica
Facultad de Farmacia Universidad de Granada, Spain
Email: jmcampos@ugr.es
Qualifications
1981 Ph.D., University of Granada, Spain
1976 B.Sc., University of Granada, Spain
Publications (selected)
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da Silva, Á.C., Scholl, J.N., de Fraga Dias, A. et al. Preclinical evaluation of bozepinib in bladder cancer cell lines: modulation of the NPP1 enzyme. Purinergic Signalling 21, 39–50 (2025). https://doi.org/10.1007/s11302-023-09975-6
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Chayah, M., Luque-González, A., Gómez-Pérez, V., Salagre, D., Al-Shdaifat, A., Campos, J. M., … Agil, A. (2024). Synthesis and Anti-Diabetic Activity of an 8-Purine Derivative as a Novel DPP-4 Inhibitor in Obese Diabetic Zücker Rats. "Drug Design, Development and Therapy, 18, 1133–1141. https://doi.org/10.2147/DDDT.S450917
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Mali SN, dos Santos CBR, Campos Rosa J and Neves Cruz J (2024) Editorial: Investigation of the biological properties of natural products using experimental approaches and in silico methods. Front. Chem. 12:1406883. doi: 10.3389/fchem.2024.1406883
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Chayah M, Luque-González A, Gómez-Pérez V, Salagre D, Al-Shdaifat A, Campos JM, Conejo-García A, Agil A. Synthesis and Anti-Diabetic Activity of an 8-Purine Derivative as a Novel DPP-4 Inhibitor in Obese Diabetic Zücker Rats. Drug Des Devel Ther. 2024;18:1133-1141 https://doi.org/10.2147/DDDT.S450917
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Campos, J., Gleitze, S., Hidalgo, C., & Núñez, M. T. (2024). IP3R-Mediated Calcium Release Promotes Ferroptotic Death in SH-SY5Y Neuroblastoma Cells. Antioxidants, 13(2), 196. https://doi.org/10.3390/antiox13020196
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Da, Vitor & Lobato, Cleison & Silva, Luciane & Santos, Igor & Barros, Elcimar & Maciel, Alexandre & Ferreira, Elenilze & Santana, Kauê & Espejo-Román, José & Campos, Joaquín & Kimani, Njogu & Santos, Cleydson. (2024). Rational Approach to New Chemical Entities with Antiproliferative Activity on Ab1 Tyrosine Kinase Encoded by the BCR-ABL Gene: An Hierarchical Biochemoinformatics Analysis. Pharmaceuticals. 1491. 10.3390/ph17111491.
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Barbosa, D. B., do Bomfim, M. R., de Oliveira, T. A., da Silva, A. M., Taranto, A. G., Cruz, J. N., de Carvalho, P. B., Campos, J. M., Santos, C. B. R., & Leite, F. H. A. (2023). Development of Potential Multi-Target Inhibitors for Human Cholinesterases and Beta-Secretase 1: A Computational Approach. Pharmaceuticals, 16(12), 1657. https://doi.org/10.3390/ph16121657
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Santos, C. B. R., Lobato, C. C., Ota, S. S. B., Silva, R. C., Bittencourt, R. C. V. S., Freitas, J. J. S., Ferreira, E. F. B., Ferreira, M. B., Silva, R. C., De Lima, A. B., Campos, J. M., Borges, R. S., & Bittencourt, J. A. H. M. (2023). Analgesic Activity of 5-Acetamido-2-Hydroxy Benzoic Acid Derivatives and an In-Vivo and In-Silico Analysis of Their Target Interactions. Pharmaceuticals, 16(11), 1584. https://doi.org/10.3390/ph16111584
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Oliveira, L. P. S., Lima, L. R., Silva, L. B., Cruz, J. N., Ramos, R. S., Lima, L. S., Cardoso, F. M. N., Silva, A. V., Rodrigues, D. P., Rodrigues, G. S., Proietti-Junior, A. A., dos Santos, G. B., Campos, J. M., & Santos, C. B. R. (2023). Hierarchical Virtual Screening of Potential New Antibiotics from Polyoxygenated Dibenzofurans against Staphylococcus aureus Strains. Pharmaceuticals, 16(10), 1430. https://doi.org/10.3390/ph16101430
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Bastos, R. S., de Lima, L. R., Neto, M. F. A., Maryam, Yousaf, N., Cruz, J. N., Campos, J. M., Kimani, N. M., Ramos, R. S., & Santos, C. B. R. (2023). Design and Identification of Inhibitors for the Spike-ACE2 Target of SARS-CoV-2. International Journal of Molecular Sciences, 24(10), 8814. https://doi.org/10.3390/ijms24108814
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Silva, L. B., Ferreira, E. F. B., Maryam, Espejo-Román, J. M., Costa, G. V., Cruz, J. V., Kimani, N. M., Costa, J. S., Bittencourt, J. A. H. M., Cruz, J. N., Campos, J. M., & Santos, C. B. R. (2023). Galantamine Based Novel Acetylcholinesterase Enzyme Inhibitors: A Molecular Modeling Design Approach. Molecules, 28(3), 1035. https://doi.org/10.3390/molecules28031035
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de Almeida, R. B. M., Barbosa, D. B., do Bomfim, M. R., Amparo, J. A. O., Andrade, B. S., Costa, S. L., Campos, J. M., Cruz, J. N., Santos, C. B. R., Leite, F. H. A., & Botura, M. B. (2023). Identification of a Novel Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase: In Vitro and In Silico Studies. Pharmaceuticals, 16(1), 95. https://doi.org/10.3390/ph16010095
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Neto, M. F. A., Campos, J. M., Cerqueira, A. P. M., de Lima, L. R., Da Costa, G. V., Ramos, R. D. S., Junior, J. T. M., Santos, C. B. R., & Leite, F. H. A. (2022). Hierarchical Virtual Screening and Binding Free Energy Prediction of Potential Modulators of Aedes Aegypti Odorant-Binding Protein 1. Molecules, 27(20), 6777. https://doi.org/10.3390/molecules27206777
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Da Costa, G. V., Neto, M. F. A., Da Silva, A. K. P., De Sá, E. M. F., Cancela, L. C. F., Vega, J. S., Lobato, C. M., Zuliani, J. P., Espejo-Román, J. M., Campos, J. M., Leite, F. H. A., & Santos, C. B. R. (2022). Identification of Potential Insect Growth Inhibitor against Aedes aegypti: A Bioinformatics Approach. International Journal of Molecular Sciences, 23(15), 8218. https://doi.org/10.3390/ijms23158218
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Silva, R. C., Freitas, H. F., Campos, J. M., Kimani, N. M., Silva, C. H. T. P., Borges, R. S., Pita, S. S. R., & Santos, C. B. R. (2021). Natural Products-Based Drug Design against SARS-CoV-2 Mpro 3CLpro. International Journal of Molecular Sciences, 22(21), 11739. https://doi.org/10.3390/ijms222111739
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Fraga Dias, A. de, Dallemole, D. R., Bruinsmann, F. A., Lopes Silva, L. F., Cruz-López, O., Conejo-García, A., … Figueiró, F. (2021). Development of Bozepinib-Loaded Nanocapsules for Nose-To-Brain Delivery: Preclinical Evaluation in Glioblastoma. Nanomedicine, 16(23), 2095–2115. https://doi.org/10.2217/nnm-2021-0164
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Santos, C. B. R., Santos, K. L. B., Cruz, J. N., Leite, F. H. A., Borges, R. S., Taft, C. A., … Silva, C. H. T. P. (2020). Molecular modeling approaches of selective adenosine receptor type 2A agonists as potential anti-inflammatory drugs. Journal of Biomolecular Structure and Dynamics, 39(9), 3115–3127. https://doi.org/10.1080/07391102.2020.1761878
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Lacal, J.C.; Zimmerman, T.; Campos, J.M. Choline Kinase: An Unexpected Journey for a Precision Medicine Strategy in Human Diseases. Pharmaceutics 2021, 13, 788. [https://10.3390/pharmaceutics13060788]
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Lacal, J. C., Zimmerman, T., & Campos, J. M. (2021). Choline Kinase: An Unexpected Journey for a Precision Medicine Strategy in Human Diseases. Pharmaceutics, 13(6), 788. https://doi.org/10.3390/pharmaceutics13060788
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Macêdo, W.J.C. et al. (2021). High-Throughput-Based Virtual Screening via Molecular Docking for Oxidative Stress Mediated by ROS Enzyme. In: La Porta, F.A., Taft, C.A. (eds) Functional Properties of Advanced Engineering Materials and Biomolecules. Engineering Materials. Springer, Cham. https://doi.org/10.1007/978-3-030-62226-8_17
Profile Details
https://www.ugr.es/en/staff/joaquin-maria-campos-rosa