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Xue, C.B., Chen, L.H., Cao, G.F., Zhang, K., Wang, A.L., Meloni, D., et al. (2010) Discovery of INCB9471, a Potent, Selective, and Orally Bioavailable CCR5 Antagonist with Potent Anti-HIV-1 Activity. Acs Medicinal Chemistry Letters, 1, 483-487.
https://doi.org/10.1021/ml1001536
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