Modelling One-Pot Method for Synthesis of 2,3-Dihydro-1H-pyrrolo[2,1-c][1,4]benzothiazine 5,5-Dioxides and Their Homologues - International Journal of Organic Chemistry

IJOC > Vol.3 No.2, June 2013

International Journal of Organic Chemistry

Volume 3, Issue 2 (June 2013)

ISSN Print: 2161-4687 ISSN Online: 2161-4695

Google-based Impact Factor: 1.26 Citations

Modelling One-Pot Method for Synthesis of 2,3-Dihydro-1H-pyrrolo[2,1-c][1,4]benzothiazine 5,5-Dioxides and Their Homologues ()

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DOI: 10.4236/ijoc.2013.32014 4,577 Downloads 7,633 Views Citations

Author(s)

Oleksandr Yu Grevtsov, Oleg V. Zaremba, Anna B. Bondarenko, Oleksandr G. Drushlyak, Sergiy M. Kovalenko, Valentyn P. Chernykh

Affiliation(s)

National University of Pharmacy, Kharkiv, Ukraine.

ABSTRACT

A facile method for synthesis of 2,3-dihydro-1H-pyrrolo[2,1-c][1,4]benzothiazines by interaction of methylenactive (2-fluorophenyl)sulfones with homologues of either 5-methoxy-3,4-dihydro-2H-pyrrole or 5-(methylthio)-3,4-dihydro- 2H-pyrrole has been developed.

KEYWORDS

Sulfones; Lactims; Cyclization; Heterocycles; Nucleophilic Aromatic Substitution

Share and Cite:

Grevtsov, O. , Zaremba, O. , Bondarenko, A. , Drushlyak, O. , Kovalenko, S. and Chernykh, V. (2013) Modelling One-Pot Method for Synthesis of 2,3-Dihydro-1H-pyrrolo[2,1-c][1,4]benzothiazine 5,5-Dioxides and Their Homologues. International Journal of Organic Chemistry, 3, 125-135. doi: 10.4236/ijoc.2013.32014.

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